Product name | Cas no | Structure | Notes |
5-Nitroisophthalic acid | 618-88-2 | ??? | Intermediate of Iohexol
|
Dimethyl 5-nitroisophthalate
| 13290-96-5 |
| Intermediate of Iohexol |
5-Amino-N,N'-bis(2,3-dihydroxypropyl) isophthaldiamide | 76820-35-4 |
| Intermediate of Iohexol |
5-Amino-N,N'-bis(2,3-dihydroxypropyl)-2,4,6-triiodo-1,3-benzenedicarboxamide | 76801-93-9 |
| Intermediate of Iohexol |
5-(Acetamido)-N,N'-bis(2,3-dihydroxypropyl)-2,4,6-triiono-1,3-benzenedicarboxamide | 31127-80-7 |
| Intermediate of Iohexol |
5-Amino-2,4,6-triiodisophthaloyl acid dichloride | 37441-29-5 |
| Intermediate of Iopamidol |
Acetoxyacetyl chloride | 13831-31-7 |
| Intermediate of contrast mediate |
(S)-(-)-2-ACETOXYPROPIONYL CHLORIDE | 36394-75-9
|
| Intermediate of contrast mediate |
Methoxyacetyl chloride | 38870-89-2 |
| Intermediate of contrast mediate |
2-Amino-1,3-propanediol | 534-03-2 |
| Intermediate of contrast mediate |
2-Amino-1,3-propanediol | 534-03-2 |
| Intermediate of contrast mediate |
4-Carboxy-5,8,11-tris(carboxymethyl)-1-phenyl-2-oxa-5,8,11-triazatridecan-13-oic acid [BOPTA] | 113786-33-7 | Gadoterate contrast mediate intermediates | |
1,4,7,10-tetraazacyclododecane base [TAZA BASE] | 294-90-6 | Gadoterate contrast mediate intermediates | |
(1,4,7,10-tetra-carboxymethyl-1,4,7,10-tetraaza-cyclododec-1-yl)-acetic acid [TAZA ACID / DOTA]
| 60239-18-1 | Gadoterate contrast mediate intermediates |
Bis(4-hydroxyphenyl) Sulfone 80-09-1 Intermediate for dyestuffs
Item No. | APIS | Intermediates |
DJ-001 | Abiraterone CAS:154229-19-3 | 1) Pyridine, 3-(diethylboryl)- CAS: 89878-14-8 2) Dehydroepiandrosterone CAS: 53-43-0 3) 17-Iodoandrosta-5,16-dien-3beta-ol CAS: 32138-69-5 4) 17-Iodoandrosta-5,16-dien-3beta-acetate ester CAS:114611-53-9 5) Androsta-5,16-diene-3,17-diol, 3-acetate17-(trifluoromethane sulfonate), (3b)- CAS:115375-60-5 |
DJ-002 |
Anamorelin CAS:249921-19-5 | 1) AnaMorelin (FuMarate) CAS: 339539-92-3 2) AnaMorelin (hydrochloride) CAS: 861998-00-7 3) tert-butyl(1-(((R)-1-((R)-3-benzyl-3-(1,2,2- trimethyl hydrazinecarbonyl) piperidin-1-yl)-3-(1H-indol-3-yl)-1- oxopropan-2-yl)amino)-2-methyl-1- oxopropan-2-yl)carbamate CAS: 339539-90-1 4) (3R)-3-Benzyl-piperidine-3-carboxylic acid triMethylhydrazide Hydrochloride CAS: 339539-84-3 5) D-Tryptophan, N-[N-[(1,1-dimethylethoxy)carbonyl]-2- methylalanyl]- CAS: 159634-94-3 6) D-Tryptophan, N-[(1,1-diMethylethoxy)carbonyl]-2-Methylalanyl-, Methyl ester CAS: 185056-99-9 7) D-Tryptophan methyl ester hydrochloride CAS: 14907-27-8 8) Ethyl (S)-3-benzylpiperidine-3-carboxylate CAS: 170844-45-8 |
DJ-003 | Apixaban CAS:503612-47-3 | 1) 1-(4-iodophenyl)-3-morpholino-5,6-dihydropyridin-2(1H)-one CAS: 473927-69-4 2) 3-(4-Morpholinyl)-1-(4-nitrophenyl)-5,6-dihydro-2(1H)-pyridinone CAS: 503615-03-0 3) 1-(4-AMinophenyl)-5,6-dihydro-3-(4-Morpholinyl)-2(1h)- pyridinone CAS: 1267610-26-3 4) 5,6-Dihydro-3-(4-morpholinyl)-1-[4-(2-oxo-1- piperidinyl)phenyl]-2(1H)-pyridinone CAS: 545445-44-1 5) 1-(4-Methoxyphenyl)-7-oxo-6-[4-(2-oxopiperidin-1- yl)phenyl]-4,5,6,7- tetrahydro-1H-pyrazolo[3,4-c]pyridine-3- carboxylic acid ethyl ester CAS: 503614-91-3 6) 4,5,6,7-Tetrahydro-1-(4-methoxyphenyl)-6-(4-nitrophenyl)-7- oxo-1H-pyrazolo[3,4-c]pyridine-3-carboxylic acid ethyl ester CAS: 536759-91-8 7) Ethyl chloro[(4-methoxyphenyl)hydrazono]acetate CAS: 27143-07-3 |
DJ-004 |
Apremilast CAS:608141-41-9 | 1) N-(1,3-dioxo-1,3-dihydroisobenzofuran-4-yl)acetamide CAS: 6296-53-3 2) 1-(3-ethoxy-4-methoxyphenyl)-2-(methylsulfonyl)ethanamine CAS: 253168-94-4 3) (S)-1-(3-Ethoxy-4-methoxyphenyl)-2-(methylsulfonyl)ethylamine N-acetyl-L-leucine salt CAS: 608141-43-1 4)(alphaS)-3-Ethoxy-4-methoxy-alpha-[(methylsulfonyl)methyl]- benzenemethanamine CAS: 608141-42-0 |
DJ-005 |
Asenapine CAS:65576-45-6 | 1) 2-(4-Chlorophenoxy)phenylacetic acid CAS: 25563-04-6 2) 5-Chloro-2-Methyl-2,3-Dihydro-Benzo-[2,3:6,7]-Oxepino- [4,5-C]-pyrrole-(2H)-One CAS: 934996-79-9 3) (5-Chloro-2-phenoxyphenyl)acetic acid CAS: 70958-20-2 4) 11-chloro-2,3-dihydro-2-methyl-1H-dibenz[2,3;6,7]oxepino[4,5- c]pyrrol-1-one CAS: 1012884-46-6 5) Trans-(+/-)-11-Chloro-2,3,3a,12b-tetrahydro-2-methyl-1H-dibenz [2,3:6,7]oxepino[4,5-c]pyrrole-1-one CAS: 129385-59-7 |
DJ-006 | Atazanavir CAS: 198904-31-3 | 1) 3,3-dimeethyl-2oxo-butanoic acid CAS: 815-17-8 2) L-tert-Leucine CAS: 20859-02-3 3) Methoxycarbonyl-L-tert-leucine CAS: 162537-11-3 |
DJ-007 | Axitinib CAS:319460-85-0 | 1) 6-Nitroindazole CAS: 7597-18-4 2) N-methyl-2-sulfanylbenzamide CAS: 20054-45-9 |
DJ-008 | Bedaquiline CAS:843663-66-1 | 1) 3-benzyl-6-bromo-2-methoxyquinoline CAS: 654655-69-3 2) 3-(dimethylamino)-1-(naphthalen-1-yl)propan-1-one CAS: 10320-49-7 3) Bedaquiline (Mixture of DiastereoMers) CAS: 654655-80-8 4) 3-benzyl-6-bromo-2-chloroquinoline CAS: 654655-68-2 5) 3-(dimethylamino)-1-(naphthalen-1-yl)propan-1-one hydrochloride CAS: 5409-58-5 6) Bedaquiline CAS: 654653-81-3 7) Bedaquiline fumarate CAS: 845533-86-0 |
DJ-009 |
Bepotastine Beslilate CAS:190786-44-8 | 1) 4-Chlorophenyl-2-pyridinylmethanol CAS: 27652-89-7 2) 2-(chloro(4-chlorophenyl)methyl)pyridine CAS: 142404-69-1 3) ethyl 4-hydroxypiperidine-1-carboxylate CAS: 65214-82-6 4) 4-[1-(4-chlorophenyl)-1-(2-pyridyl)methoxy]piperidine CAS: 122368-54-1 5) (s)-4-[1-(4-chlorophenyl)-1-(2-pyridyl)methoxy]piperidine CAS: 201594-84-5 |
DJ-010 | Bezafibrat CAS:41859-67-0 |
|
DJ-011 | Bosentan CAS:147536-97-8 | 1) 2-Cyanopyrimidine CAS: 14080-23-0 2) 4,6-Dichloro-5-(2-methoxyphwnoxy)-2 ,2’-bipyrimidine CAS: 150728-13-5 3) 4-tert-Butyl-N-(6-chloro-5-(2-methoxyphenoxy)-2,2’-bipyrimidin- 4-yl)benzenesulfonamide CAS: 150727-06-3 |
DJ-012 |
Canagliflozin CAS:842133-18-0 | 1) (3R,4S,5R,6R)-3,4,5-tris(triMethylsilyloxy)-6- ((triMethylsilyloxy)Methyl)tetrahydro-2H-pyran-2-one CAS: 32384-65-9 2) 2-(5-BroMo-2-Methylbenzyl)-5-(4-fluorophenyl)thiophene CAS: 1030825-20-7 3) 2-(4-Fluorophenyl)-5-[(5-iodo-2-methylphenyl)methyl]thiophene CAS: 898566-17-1 |
DJ-013 | Carfilzomib* CAS:868540-17-4 | 1) (S)-2-amino-4-methyl-1-((R)-2-methyloxiran-2-yl)pentan-1-one CAS: 247068-85-5 2) 4-Morpholine acetic acid hydrochloride CAS: 89531-58-8 3) (S)-2-((S)-4-methyl-2-((S)-2-(2-morpholinoacetamido)-4 -phenylbutanamido)pentanamido)-3-phenylpropanoic acid CAS: 868540-16-3 4) (S)-tert-butyl (2,6-dimethyl-3-oxohept-1-en-4-yl)carbamate CAS: 247068-81-1 5) tert-butyl ((S)-4-methyl-1-((R)-2-methyloxiran-2-yl)-1- oxopentan-2-yl)carbamate CAS: 247068-82-2 6) (S)-2-amino-4-methyl-1-((R)-2-methyloxiran-2-yl)pentan-1-one CAS: 247068-84-4 7) (S)-methyl 2-((S)-2-((S)-2-amino-4-phenylbutanamido)-4-methyl pentanamido)-3-phenylpropanoate CAS: 868539-98-4 8) (S)-methyl 2-((S)-2-((S)-2-amino-4-phenylbutanamido)-4-methyl pentanamido)-3-phenylpropanoate trifluoroacetate CAS: 868539-99-5 9) 4-Morpholine acetic acid CAS: 3235-69-6
|
DJ-014 |
CAS:1032900-25-6 | 1) tert-butyl 4-(4-amino-5-isopropoxy-2-methylphenyl)piperidine- 1-carboxylate CAS: 1032903-63-1 2) 2,5-dichloro-N-(2-(isopropylsulfonyl)phenyl)pyrimidin-4-amine CAS: 761440-16-8 3) 1-chloro-5-fluoro-2-methyl-4-nitrobenzene CAS: 112108-73-3 4) 1-chloro-5-isopropoxy-2-methyl-4-nitrobenzene CAS: 1032903-50-6 5) 2-isopropoxy-5-methyl-4-(piperidin-4-yl)aniline CAS: 1380575-45-0 6) 2-isopropoxy-5-methyl-4-(piperidin-4-yl)aniline CAS: 1035230-24-0 7) tert-butyl 4-(4-((5-chloro-4-((2-(isopropylsulfonyl)phenyl)amino) pyrimidin-2-yl)amino)-5-isopropoxy-2-methylphenyl)piperidine- 1-carboxylate CAS: 1032903-64-2 8) 2-(isopropylsulfonyl)aniline CAS: 76697-50-2 |
DJ-015 |
Cinacalcet CAS:226256-56-0 | 1) 3-(trifluoromethyl)cinnamic acid CAS: 779-89-5 2) 3-(3-Trifluoromethylphenyl)propionic acid CAS: 585-50-2 3) 3-(Trifluoromethyl)benzenepropanol CAS: 78573-45-2 4) 3-(3-Trifluoromethylphenyl)propionaldehyde CAS: 21172-41-8 5) R-(+)-alpha-(1-Naphthyl)ethylamine CAS: 3886-70-2 6) (S)-(+)-1-(1-Naphthyl)ethylamine CAS: 10420-89-0 |
DJ-016 |
Darifenacin HBr CAS:133099-07-7 | 1) (S)-2,2-diphenyl-2-(pyrrolidin-3-yl)acetonitrile hydrobromide CAS: 194602-27-2 2) (S)-Alpha,Alpha-Diphenyl-3-pyrrolidine acetamide L-Tartaric acid salt CAS: 134002-26-9 3) 5-(2-bromoethyl)octahydrobenzofuran CAS: 127264-14-6 |
DJ-017 |
Dapagliflozin CAS:461432-26-8 | 1) (5-bromo-2-chlorophenyl)(4-ethoxyphenyl)methanone CAS: 461432-22-4 2) 5-bromo-2-chloro-4’-ethoxydiphenylmethane CAS: 461432-23-5 |
DJ-018 |
Dronedarone HCl CAS:141625-93-6 | 1) N-(3-Chloropropyl)dibutylamine CAS: 36421-15-5 2) 2-N-butyl-5-nitrobenzofuran CAS: 133238-87-6 3) 2-butyl-3-(4-hydroxybenzoyl)-5-nitrobenzofuran CAS: 141645-16-1 4) 2-Butyl-3-(4-(3-dibutylaminopropoxy)benzoyl)-5-Nitrobenzofuran CAS: 141645-23-0 5) 4-[3-(Dibutylamino)propoxy]benzoic acid hydrochloride CAS: 437651-44-0 6) 2-Butyl-5-[methanesulfonamido]benzofuran CAS: 437652-07-8 7) (5-amino-2-butylbenzofuran-3-yl)(4-(3-(dibutylamino)propoxy) phenyl)methanone dioxalate CAS: 500791-70-8 |
DJ-019 |
Eletriptan HBr CAS:177834-92-3 | 1) 5-Bromoindole CAS: 10075-50-0 2) 5-bromo-3-[1-methylpyrrolidin-2(R)-ylmethyl]indole CAS: 143322-57-0 3) Phenyl vinyl sulfone CAS: 5535- 48- 8 4) 1-acetyl-5-bromo-3-{[(2R)-1-methylpyrrolidin-2-yl]methyl}-1H- indole CAS: 205369-12-6 5) Ethanone,1-[3-[[(2R)-1-methyl-2-pyrrolidinyl]methyl]-5-[(1E)-2- (phenylsulfonyl)ethenyl]-1H-indol-1-yl]- CAS: 188113-71-5 |
DJ-020 |
Favipiravir CAS:259793-96-9 | 1) 6-bromo-3-hydroxypyrazine-2-carboxamide CAS: 259793-88-9 2) 3,6-dichloropyrazine-2-carbonitrile CAS: 356783-16-9 3) 3,6-difluoropyrazine-2-carbonitrile CAS: 356783-28-3 |
DJ-021 |
Fesoterodine CAS:286930-02-7 | 1) 3-[3-[Bis(1-methylethyl)amino]-1-phenylpropyl]-4-hydroxy Benzenemethanol CAS: 200801-70-3 2) 3-[(1R)-3-[Bis(1-methylethyl)amino]-1-phenylpropyl]-4- Hydroxybenzenemethanol CAS: 207679-81-0 |
DJ-022 | Ganciclovir CAS:82410-32-0 | 1) Triacetylganciclovir CAS: 86357-14-4 2) 1,3-Diacetoxy-2-(acetoxymethoxy)propane CAS: 86357-13-3 |
DJ-023 |
Ibrutinib* CAS:936563-96-1 | 1) 3-(4-phenoxyphenyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine CAS: 330786-24-8. 2) (R)-3-(4-phenoxyphenyl)-1-(piperidin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine CAS: 1022150-12-4 3) (S)-1-Boc-3-hydroxypiperidine CAS: 143900-44-1 4) 1-iodo-4-phenoxybenzene CAS: 2974-94-9 5) 1-bromo-4-phenoxybenzene CAS: 101-55-3 6) 4-phenoxyphenylboronic acid CAS: 51067-38-0 7) 1H-pyrazolo[3,4-d]pyrimidin-4-amine CAS: 2380-63-4 8) 3-iodo-1H-pyrazolo[3,4-d]pyrimidin-4-amine CAS: 151266-23-8 9) 5-amino-1H-pyrazole-4-carbonitrile CAS: 16617-46-2 |
DJ-024 |
LCZ696* Valsartan/sacubitril (1:1) CAS:936623-90-4 | 1) (R,E)-5-([1,1'-biphenyl]-4-yl)-4-((tert-butoxycarbonyl)amino)- 2-methylpent-2-enoic acid CAS: 1012341-48-8 2) (2R,4S)-5-([1,1'-biphenyl]-4-yl)-4-((tert-butoxycarbonyl)amino)- 2-methylpentanoic acid CAS: 1012341-50-2 3) (2R,4S)-ethyl 5-([1,1'-biphenyl]-4-yl)-4-amino- 2-methylpentanoate hydrochloride CAS: 149690-12-0 4) (R)-3-([1,1'-biphenyl]-4-yl)-2-aminopropanoic acid CAS: 170080-13-4 5) AHU-377 (heMicalciuM salt) CAS: 1369773-39-6 6) 5-([1,1'-biphenyl]-4-yl)-4-((tert-butoxycarbonyl)aMino)-2- Methylpentanoate CAS: 149709-60-4 7) AHU-377 CAS: 149709-62-6 |
DJ-025 |
CAS:1441674-54-9 | 1) (6S)-5-Azaspiro[2.4]heptane-5,6-dicarboxylic acid 5- (1,1-dimethylethyl) ester potassium salt (1:1) CAS: 1441673-92-2 2) 1-(7-broMo-9,9-difluoro-9H-fluoren-2-yl)-2-chloro-Ethanone CAS: 1378387-81-5 3) 2-Azabicyclo[2.2.1]heptane-2-carboxylic acid 3-(6-bromo-1H- benzimidazol-2-yl)-,1,1-dimethylethylester, (1R,3S,4S) CAS: 1256387-74-2 |
DJ-026 |
Linagliptin CAS:668270-12-0 | 1)2-(chloromethyl)-4-methylquinazoline CAS: 109113-72-6 2)8-Bromo-3-methyl-1H-purine-2,6(3H,7H)-dione CAS: 93703-24-3 3)(R)-3-(Boc-Amino)piperidine CAS: 309956-78-3 4)1-Bromobut-2-yne CAS: 3355-28-0 |
DJ-027 | Linezolid CAS:165800-03-3 | 1) (S)-(+)-Glycidyl phthalimide CAS: 161596-47-0 2) 3-Fluoro-4-morpholin-4-yl-phenylamine CAS: 93246-53-8 3) (S)-N-[[3-[3-Fluoro-4-(4-morpholinyl)phenyl]-2-oxo-5-oxazolidinyl] phthalimide CAS: 168828-89-5 |
DJ-028 | Lorcaserin CAS: 616202-92-7 | 1) 1-[[2-(4-Chlorophenyl)ethyl]amino]-2-chloropropane CAS: 953789-37-2 2) LorcaserinA CAS: 616201-80-0
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DJ-029 |
CAS:936727-05-8 | 1) 3-(6-Amino-3-methyl-pyridin-2-yl)-benzoicacidtert-butylester CAS: 1083057-14-0 2) 1-(2,2-Difluoro-benzo[1,3]dioxol-5-yl)-cyclopropanecarboxylicacid CAS: 862574-88-7
|
DJ-030 |
CAS: 441798-33-0 | 1) 5-(4-broMophenyl)-4,6-dichloro-PyriMidine CAS: 146533-41-7 2) N-Propyl-sulfamide potassium salt CAS: 1393813-41-6 3) N-Propyl-sulfamide potassium CAS: 147962-41-2 |
DJ-031 | Mycophenolate mofetil CAS:128794-94-5 | 1) MYCOPHENOLATE SODIUM CAS: 37415-62-6
|
DJ-032 |
CAS:698387-09-6 | 1) 6-amino-4-(3-chloro-4-(pyridin-2-ylmethoxy)phenylamino)-7- ethoxyquinoline-3-carbonitrile CAS: 848139-78-6 2) 4-Chloro-3-cyano-7-ethoxy-6-nitroquinoline CAS: 214476-09-2 3) 3-chloro-4-(pyridin-2-ylmethoxy)aniline CAS: 524955-09-7 |
DJ-033 |
CAS:656247-18-6 | 1) Nintedanib CAS: 656247-17-5 2) N-(4-aminophenyl)-N-methyl-2-(4-methylpiperazin-1-yl)acetamide CAS: 262368-30-9 3) methyl 2-oxoindoline-6-carboxylate CAS: 14192-26-8 4) (E)-methyl 3-(methoxy(phenyl)methylene)-2-oxoindoline-6-carboxylate CAS: 1168150-46-6 |
DJ-034 |
CAS:603139-19-1 | 1) L-Leucine, 4-fluoro-, ethyl ester, sulfate (1:1) CAS: 848949-85-9 2) 2,2,2-trifluoro-1-(4'-(Methylsulfonyl)biphenyl-4-yl)ethanone CAS: 893407-18-6 3) 1-Amino-1-cyclopropanecarbonitrile hydrochloride CAS: 127946-77-4 |
DJ-035 | Omarigliptin* CAS:1226781-44-7 | 1) 2-(Methylsulfonyl)-2,4,5,6-tetrahydropyrrolo[3,4-c]pyrazole CAS: 1280210-80-1 2) tert-butyl (1-(methoxy(methyl)amino)-1-oxopent-4-yn-2-yl)carbamate CAS: 1172623-95-8 3) tert-butyl [(2R,3S)-2-(2,5-difluorophenyl)-5-oxotetrahydro-2H-pvran -3 yl]carbamate CAS: 951127-25-6 4) 2-(Methylsulfonyl)-2,4,5,6-tetrahydropyrrolo[3,4-c]pyrazole CAS: 1280210-80-1 |
DJ-036 |
Palbociclib* CAS:571190-30-2 | 1) 2-chloro-8-cyclopentyl-5-methylpyrido[2,3-d]pyrimidin-7(8H)-one CAS: 1013916-37-4 2) 6-bromo-2-chloro-8-cyclopentyl-5-methylpyrido[2,3-d]pyrimidin-7(8H) -one CAS: 1016636-76-2 3) tert-butyl 4-(6-nitropyridin-3-yl)piperazine-1-carboxylate CAS: 571189-16-7 4) tert-butyl 4-(6-aminopyridin-3-yl)piperazine-1-carboxylate CAS: 571188-59-5 5) 5-bromo-2,4-dichloropyrimidine CAS: 36082-50-5 6) 5-bromo-2-chloro-N-cyclopentylpyrimidin-4-amine CAS: 733039-20-8 |
DJ-037 | Pazopanib CAS:444731-52-6 | 1) 2,3-Dimethyl-6-amino-2H-indazole (dihydrochloride) NO CAS. 2) 2,4-Dichloropyrimidine CAS: 3934-20-1 3) 3-Methyl-6-nitroindazole CAS: 6494-19-5 |
DJ-038 | Posaconazole CAS:171228-49-2 | 1) 1-((2S,3S)-2-(benzyloxy)pentan-3-yl)-4-(4-(4-(4-hydroxyphenyl) piperazin-1-yl)phenyl)-1H-1,2,4-triazol-5(4H)-one CAS: 184177-83-1 2) ((3S,5R)-5-((1H-1,2,4-triazol-1-yl)methyl)-5-(2,4-difluorophenyl)tetrahy drofuran-3-yl)methyl 4-methylbenzenesulfonate CAS: 149809-43-8 |
DJ-039 |
Pralatrexate CAS:146464-95-1 | 1) 6-Bromomethyl-pteridine-2,4-diamine hydrobromide CAS: 52853-40-4 2) Benzeneacetic acid, 4-(methoxycarbonyl)-,methyl ester CAS: 52787-14-1 3) Benzeneacetic acid,4-(methoxycarbonyl)-.alpha.-2-propyn-1-yl-, methyl ester CAS: 146464-90-6 4) 2,4-diamino-.alpha.-(4-carboxyphenyl) -.alpha.-2-propyn-1-yl -6-Pteridinepropanoic acid CAS: 146464-92-8 5) Benzoic acid, 4-[1-[(2,4-diamino-6-pteridinyl)methyl]-3-butyn-1-yl]- CAS: 146464-93-9 |
DJ-040 | Propiverine Hydrochloride CAS:54556-98-8 |
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DJ-041 | Ramelteon CAS:196597-26-9 | 1) 1,2,6,7-Tetrahydro-8H-indeno[5,4-b]furan-8-one CAS: 196597-78-1 2) (E)-2-(6,7-dihydro-1H-indeno[5,4-b]furan-8(2H)-ylidene)acetonitrile CAS: 196597-79-2 3) 1,6,7,8-Tetrahydro-2H-indeno[5,4-b]furan-8-ethanamine hydrochloride CAS: 1053239-39-6 4) (S)-2-(1,6,7,8-Tetrahydro-2H-indeno[5,4-b]furan-8-yl)ethylamine Hydrochloride CAS: 196597-80-5 |
DJ-042 |
Regorafenib CAS:755037-03-7 | 1) 1-chloro-4-isocyanato-2-(trifluoromethyl)benzene CAS: 327-78-6 2) 4-amino-3-fluorophenol CAS: 399-95-1 3) 4-chloro-N-methylpicolinamide CAS: 220000-87-3 4) 4-(4-amino-3-fluorophenoxy)-N-methylpyridine-2-carboxamide CAS: 757251-39-1 |
DJ-043 |
Rivaroxaban CAS:366789-02-8 | 1) 2-[(2S)-oxiran-2ylmethyl]-1H-isoindole-1,3(2H)-dione CAS:161596-47-0 2) 4-(4-aminophenyl)morpholin-3-one CAS: 438056-69-0 3) 5-Chlorothiophene-2-carboxylic acid CAS: 24065-33-6 4) 5- Chlorothiophene-2-carbonyl chloride CAS: 42518-98-9, 5) (S)-4-(4-(5-(Aminomethyl)-2-oxooxazolidin-3-yl)phenyl)morpholin-3- one hydrocloride CAS: 898543-06-1 |
DJ-044 | Rotigotine HCl CAS:125572-93-2 | 1) 5-methoxy-2-tetralone CAS: 32940-15-1 2) (S)-5-methoxy-1,2,3,4-tetrahydronaphthalen-2-amine CAS: 105086-80-4 3) (S)-5-methoxy-1,2,3,4-tetrahydronaphthalen-2-amine hydrochloride CAS: 58349-17-0 4) (S)-1,2,3,4-Tetrahydro-5-methoxy-N-propyl-2-naphthalenamine hydrochloride CAS: 93601-86-6 5) (S)-5-methoxy-N-propyl-N-(2-(thiophen-2-yl)ethyl)-1,2,3,4- tetrahydronaphthalen-2-amine CAS: 101945-65-7 |
DJ-045 | Saxagliptin CAS: 361442-04-8 | 1) 3-Hydroxy-1-adaMantyl-D-glycine CAS: 709031-29-8 |
DJ-046 | Selexipag CAS:475086-01-2 | 1) 5-chloro-2,3-diphenylpyrazine CAS: 41270-66-0 2) 4-(Isopropylamino)butanol CAS: 42042-71-7 3) 1-Butanol, 4-[(5,6-diphenylpyrazinyl)(1-methylethyl)amino]- CAS: 475086-75-0
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DJ-047 |
Silodosin CAS:160970-54-7 | 1) 2-[2-(2,2,2-Trifluoroethoxy)phenoxy]ethyl methanesulfonate CAS: 160969-03-9 2) 5-[(2R)-2-Aminopropyl]-1-[3-(benzoyloxy)propyl]-2,3-dihydro-1H-indole-7-carbonitrile(2R,3R)-2,3-dihydroxybutanedioate CAS: 239463-85-5 |
DJ-048 |
Sofosbuvir CAS:1190307-88-0 | 1) Cytidine, N-benzoyl-2'-deoxy-2'-fluoro-2'-methyl-, 3',5'-dibenzoate,(2'R)-CAS: 817204-32-3 2) 2-C-methyl-4,5-O-(1-methylethylidene)-,ethyl este CAS: 93635-76-8 3) ((2R,3R,4R)-3-(benzoyloxy)-4-fluoro-4-methyl-5-oxotetrahydrofuran-2-yl)methyl benzoate CAS: 874638-80-9 4) 2'-deoxy-2'-fluoro-2'-C-methyluridine CAS: 863329-66-2 5) 2'-deoxy-2'-fluoro-2'-C-methylcytidine CAS: 817204-33-4 6) N-[(S)-(2,3,4,5,6-Pentafluorophenoxy)phenoxyphosphinyl]-L- alanine 1-methylethyl ester CAS: 1334513-02-8 |
DJ-049 | Suvorexant CAS:1030377-33-3 | 1) (R)-5-chloro-2-(5-methyl-1,4-diazepan-1-yl)benzo[d]oxazoleCAS: 1266975-27-2 2) 5-methyl-2-(2H-1,2,3-triazol-2-yl)benzoic acid CAS: 956317-36-5 3) (R)-4-(5-chlorobenzo[d]oxazol-2-yl)-7-Methyl-1,4-diazepan-1-iuM (2S,3S)-2,3-bis(benzoyloxy)-3carboxypropanoate CAS:1276666-14-8 4) 5-Chlorobenzooxazole-2-thiol CAS: 22876-19-3 5) tert-butyl 2-(5-chlorobenzo[d]oxazol-2-ylaMino)ethylcarbaMate CAS: 1144509-75-0 |
DJ-050 | Tadalafil CAS:171596-29-5 | 1) N-Acetyl-L-Tryptophan CAS: 1218-34-4 2) N-Acetyl-DL-tryptophan CAS: 87-32-1 3) D-Tryptophan CAS: 153-94-6 4) D-Tryptophan methyl ester Hcl CAS: 14907-27-8 5) Tadalafil CIS intermediate CAS: 171752-68-4 6) Chloro acetyl carbolines CAS: 171489-59-1 |
DJ-051 | Tasquinimod CAS:254964-60-8 | 1) 4-hydroxy-5-methoxy-1-methyl-2-oxo-1,2-dihydroquinoline-3-carboxylicacid CAS: 248282-18-0 2) N-methyl-4-(trifluoromethyl)aniline CAS: 22864-65-9
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DJ-052 | Teneligliptin CAS:760937-92-6 | 1) (2S)-4-Oxo-2-(3-thiazolidinylcarbonyl)-1-pyrrolidinecarboxylic acidtert-butyl ester CAS: 401564-36-1 2) 1-(3-methyl-1-phenyl-1H-pyrazol-5-yl)piperazine CAS: 401566-79-8 |
DJ-053 |
Ticagrelor CAS:274693-27-5 | 1) (1R,2S)-2-(3,4-Difluorophenyl)cyclopropan aminium (2R)-hydroxy (phenyl)Ethanoate CAS: 376608-71-8 2) (1R,2S)-2-(3,4-Difluorophenyl)cyclopropanaminium hydrochlorideCAS: 1402222-66-5 3) (1R,2S)-rel-2-(3,4-Difluorophenyl)cyclopropanamine hydrochlorideCAS: 1156491-10-9 4) N-[(3aS,4R,6S,6aR)-Tetrahydro-6-hydroxy-2,2-dimethyl-4H-cyclopenta-1,3-dioxol-4-yl]carbamicacid phenylmethyl ester CAS: 274693-53-7 5) 2-((3aR,4S,6R,6aS)-6-amino-2,2-dimethyltetrahydro-3aH-cyclopenta[d][1,3]dioxol-4-yloxy)ethanol L-tataric acid CAS: 376608-65-0 6) 4,6-dichloro-2-propylthiopyrimidine-5-amine CAS: 145783-15-9 7) Ethanol, 2-[[(3aR,4S,6R,6aS)-6-[[5-amino-6-chloro-2-(propylthio)-4-pyrimidinyl]amino]tetrahydro-2,2-dimethyl-4H-cyclopenta-1,3-dioxol-4-yl]oxy]- CAS: 1156491-10-9 |
DJ-054 | Tildipirosin CAS:328898-40-4 |
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DJ-055 | Tipiracil HCl CAS:183204-72-0 | 1) 6-(Hydroxymethyl)uracil CAS: 22126-44-9 2) 6-(Chloromethyl)uracil CAS: 18592-13-7 3) 3,4-Dihydro-2H-pyrrol-5-amine hydrochloride CAS: 7544-75-4 |
DJ-056 |
Tofacitinib citrate CAS:540737-29-9 | 1) 4-Chloropyrrolo[2,3-d]pyrimidine CAS: 3680-69-1 2) 4-Chloro-7-[(4-methylbenzene)sulfonyl]-7H-pyrrolo[2,3-d]pyrimidine CAS: 479633-63-1 3) 2, 4-dichloro-7H-pyrrol-(2, 3-d)pyrimidine CAS: 90213-66-4 4) (3R, 4R)-N, 4-Dimethyl-1-(phenylmethyl)-3-piperidinamine CAS: 477600-70-7 5) (3R, 4R)-N, 4-Dimethyl-1-(phenylmethyl)-3-piperidinamine hydrochloride CAS: 1062580-52-2 6) Bis[(3R,4R)-N,4-dimethyl-1-(phenylmethyl)-3-piperidinamine] di-p-toluyl-L-tartrate CAS: 477600-71-8 7) N-methyl-N-((3R,4R)-4-methylpiperidin-3-yl)-7H-pyrrolo[2,3-d] Pyrimidin-4-amine CAS: 477600-74-1 |
DJ-057 | Umeclidinium bromide CAS:869113-09-7 | 1) diphenyl(quinuclidin-4-yl)methanol CAS: 461648-39-5 |
DJ-058 |
Vilazodone CAS:163521-12-8 | 1) 3-(4-chloro-butyl)-5-cyanoindole CAS: 143612-79-7 2) 5-nitrobenzofuran-2-carboxylic acid ethyl ester CAS: 69604-00-8 3) ethyl 5-aminobenzofuran-2-carboxylate CAS: 174775-48-5 4) 1-(2-aminocarbonylbenzofuran-5-yl)piperazine CAS: 183288-46-2 |
DJ-059 | Intermediate of Ceftizoxime, Ceftibuten and Cefroxadine | 1) 7-Phenyl acetylamino-3-hydroxy-3-cephemcyclo-4-carboxylic acid diphenyl methyl ester(3-OH) CAS: 54639-48-4 |
DJ-060 | Intermediate of 5th. generation cephalosporins | 1) [Diphenylmethyl α-[3-benzyl-7-oxo-4-thia-2,6-diazabicyclo [3,2,0] hept-2-en-6-yl]-α-(1- morpholinoethylidene)](ENM) CAS: 84532-49-6 |
DJ-061 | Intermediate of Sartans type | 1) 4-Bromomethyl-2-cyanobiphenyl CAS: 114772-54-2 |
DJ-062 | Intermediate of pesticide | 1) 4-Chlorobenzotrifluoride CAS: 98-56-6 2) Benzotrifluoride CAS: 98-08-8 |